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mGluR3 Agonists

  • NMDA receptor
  • AMPA receptor
  • mGluR2
  • mGluR3
  • mGluR4
  • mGluR5
Nº Cat. Nombre del producto Información Selectivo / Pan IC50 / Ki
S6001 LY404039 LY404039 is a potent agonist of recombinant human mGlu2/mGlu3 receptors with Ki of 149 nM/92 nM, shows >100-fold selectivity over ionotropic glutamate receptors, glutamate transporters, and other receptors. Phase 3. Pan Rat neurons expressing native mGlu2/3, Ki: 88 nM; Recombinant human mGlu3, Ki: 92 nM