CYP2-Selectivo Inhibitors
- P450
- CYP2
- CYP3
- CYP1
- CYP17
| Nº Cat. | Nombre del producto | Información | Selectivo / Pan | IC50 / Ki |
|---|---|---|---|---|
| S4221 | Benzbromarone | Benzbromarone is a CYP2C9 inhibitor, it binds to CYP2C9 with Ki value of 19.3 nM. | Selective | CYP2C9, Ki: 19.3 nM |
| S2262 | Apigenin | Apigenin is a potent P450 inhibitor for CYP2C9 with Ki of 2 μM. | Selective | CYP2C9, Ki: 2 μM |
| S2268 | Baicalein | Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor. | Selective | |
| S2046 | Pioglitazone HCl | Pioglitazone HCl is a hydrochloride salt form of pioglitazone which is a cytochrome P450 (CYP)2C8 and CYP3A4 enzymes inhibitor for CYP2C8, CYP3A4 and CYP2C9 with Ki of 1.7 μM, 11.8 μM and 32.1 μM, respectively. | Pan | CYP2C9, Ki: 32.1 μM; CYP2C8, Ki: 1.7 μM |
| S2187 | Avasimibe | Avasimibe inhibits ACAT with IC50 of 3.3 μM, also inhibits human P450 isoenzymes CYP2C9, CYP1A2 and CYP2C19 with IC50 of 2.9 μM, 13.9 μM and 26.5 μM, respectively. | Pan | CYP2C19, IC50: 26.5 μM; CYP2C9, IC50: 2.9 μM |
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